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Basically, the problem for a lot of labs is that single-target peptides often hit a plateau in metabolic studies, and you need something that can pull multiple levers at once to really see what's happening with glucose and weight regulation.
What this does is it hits three receptors—GCGR, GIPR, and GLP-1R—in one shot, which is pretty much a more complete way to mimic how the body naturally handles energy balance, and we've seen it outperform older single agonists in head-to-head comparisons.
It's a, soluble in water at 5mg/ml, and you'll want to store it at -20°C where it'll stay stable for about 3 years—though we usually have stock, but confirm lead time if you need it fast. The EC50 values are 5.79 nM for GCGR, 0.0643 nM for GIPR, and 0.775 nM for GLP-1R, so it's particualrly potent on teh GIPR side.
our company offer it in 2.5mg, 5mg, 10mg, or 15mg vials, and most buyers go with the 10mg for general dosing—it's easier to reconstitute. For supply, we run GMP and ISO 9001, but this is strictly for research use only, not for human or veterinary appliction.
One thing to keep in mind is it's not ideal for acute glucose clamp studies where you need a fast-acting short pulse—its duration is longer than something like liraglutide, so plan your protocol accordingly. Also, the molecular weight is 4113.58 g/mol give or take 1.0, which means you'll need to calculate molarity carefully if you're doing receptor binding assays.
Anyway, the shelf life is solid at 3 years, and we ship with COAs, so you're not guessing about purity or activity.
We can start with as little as 10 vials per specification, but if you need smaller amounts for initial testing, just let us know and we can work something out.
For standard 2.5mg, 5mg, 10mg, and 15mg vials, we usually ship within 5-7 business days. Custom formulations might add a few extra days depending on the request.
Yes, we include a Certificate of Analysis with every order, covering purity over 99% and confirming GMP and ISO 9001 compliance. USP documentation is also available on request.
It's soluble in water at 5mg/ml and should be stored at -20°C. Under those conditions, the shelf life is 3 years from the date of manufacture.
Absolutely, we can adjust vial sizes and packaging to fit your lab's workflow. Just tell us the total quantity and any special requirements, and we'll prepare a quote.
