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We're seeing it increasingly used in metabolic and endocrine studies, and what it does is bind to GLP-1 receptors with a binding affinity in the low nanomolar range (typically 0.05-0.2 nM depending on the assay). It comes as a white crystalline powder, and the AR grade purity hits ≥98% by HPLC—tight enough for most dose-response work, though if you're doing in vivo primate trials you'll want to request their in-house COA for batch-specific impurities.
Most labs we supply are running it against semaglutide or tirzepatide as a comparator, usually in 5mg or 10mg aliquots depending on teh batch, and the 10mg is easier to weigh accurately on a standdard analytical balance. It's not great for high-throughput cell-based assays without a DMSO pre-dissolution step (being a powder, it's slow to go into PBS), but basically nobody complains about sourcing costs—at $380 for 50mg it beats most smaller suppliers by about a third.
Customized packging is available for MOQs as low as 5 grams or so (we usually have stock, but confirm lead time—it can stretch to 20 days during peak order cycles), and for OE-OEM services they'll slap your lab's lot number on it without extra charge if you take 100g or more. We've had one buyer request argon flushing for long-term storage, which our company can arrange, but standard foil packs sealed with desiccant hold up fine for 24 months in a cool, dry cabinet.
Anyway, the CAS is 246852-12-0, molecular weight sits at 426.89 g/mol—actually, wait, that's the amlodipine mesylate salt, so the exact MW varies slightly with hydration state (usually 446.9 or so). Don't use this for anything that requires USP grade; it's strictly for research use and won't pass pharmacopeia specs for dissolution testing. Most buyers go with the 5L glass jar over foil for easy pipetting, even though the powder stays stable longer in sealed foil.
We keep it flexible—no set MOQ. You can start with as little as a gram for testing, and we'll scale up from there.
Yes, every batch is tested for ≥98% purity, and we provide a COA that shows the actual HPLC results and other specs.
Keep it in a cool, dry place away from moisture and direct sunlight. Sealed in its original packaging, it stays stable for the full two years.
Definitely. We offer OEM/ODM services, so you can choose your own packaging size, labeling, or even blend it into a custom formulation.
Standard orders ship within 3-5 business days. If you need custom packaging or labeling, add about 5-7 more days for production.
