We've been getting a lot of requests for something that hits all three receptors without needing to mix compounds, and this one does it—GCGR at 5.79 nM, GIPR at 0.0643 nM, and GLP-1R at 0.775 nM, which is pretty much the sweet spot for metabolic studies. It's a white crystalline or lyophilized powder, 4.6 kDa roughly, and purity runs ≥99% by HPLC with peptide content above 92%.
Most buyers go with teh 5mg or 10mg vials for dosing flexibility, though we also stock 2mg, 100mg, 1g, and 10g if you're scaling up. You'll want to store it at 2-8°C and keep it out of light—it's soluble in DMSO, so reconstitution is straightforward.
What it does is target obesity and type 2 diabetes pathways, but it's not suited for anything beyond research purposes. We usually have stock on smaller sizes, but the 10g vials can take 20 days or so to ship (confirm lead time).
One thing you might not think to ask: the lyophilized form can be a bit hygroscopic, so open it in a dry enviroment. Also, the EC50 values we quote are for human receptors, so if you're working with animal models, expect some variance.
GMP compliant production, and we'll include a COA with every batch. The 100mg vial is actually easier to handle for larger runs than multiple 10mg ones—fewer vials to reconstitute.
Anyway, that's the gist of it. No need to overcomplicate the ordering—just pick your vial size and we'll get it out.
Standard lead time is 7–14 business days for stock sizes like 10g. If you need a rush order, let us know and we can often speed that up.
Yes, each batch is HPLC-verified and comes with a Certificate of Analysis showing the ≥99% purity. You'll get it with your shipment.
We can do custom vial sizes for bulk orders—just reach out with your required quantity. For smaller research needs, the standard options cover most cases.
Keep it at 2–8°C in a fridge, away from direct light. Sealed vials stored this way stay stable for up to 24 months.
We supply a GMP compliance statement along with the COA. If you need additional batch records or a full quality dossier, that can be arranged per request.